Dr. Yousaf Khan

I am a Chemist by professional and specializing in Organic Chemistry Medicinal Chemistry Green Chemistry, with expertise in Drug designing, drug synthesis, drug development

Structure-guided optimization of N-(5-((2-oxopropyl) thio)-1, 3, 4-thiadiazol-2-yl) propionamide frameworks as potent SARS-CoV-2 Mpro inhibitor for treating coronavirus disease


Journal article


Maher S Alwethaynani, Reem Nabil Hassan, Rafaqat Hussain, Hina Sarfraz, Asma Sardar, Faisal Asif, Yousaf Khan, Ammena Y Binsaleh, Nawal Al-Hoshani, Mariam Ameen Mojally, others
Bioorganic Chemistry, Elsevier, 2026, p. 110102

Cite

Cite

APA   Click to copy
Alwethaynani, M. S., Hassan, R. N., Hussain, R., Sarfraz, H., Sardar, A., Asif, F., … others. (2026). Structure-guided optimization of N-(5-((2-oxopropyl) thio)-1, 3, 4-thiadiazol-2-yl) propionamide frameworks as potent SARS-CoV-2 Mpro inhibitor for treating coronavirus disease. Bioorganic Chemistry, 110102.


Chicago/Turabian   Click to copy
Alwethaynani, Maher S, Reem Nabil Hassan, Rafaqat Hussain, Hina Sarfraz, Asma Sardar, Faisal Asif, Yousaf Khan, et al. “Structure-Guided Optimization of N-(5-((2-Oxopropyl) Thio)-1, 3, 4-Thiadiazol-2-Yl) Propionamide Frameworks as Potent SARS-CoV-2 Mpro Inhibitor for Treating Coronavirus Disease.” Bioorganic Chemistry (2026): 110102.


MLA   Click to copy
Alwethaynani, Maher S., et al. “Structure-Guided Optimization of N-(5-((2-Oxopropyl) Thio)-1, 3, 4-Thiadiazol-2-Yl) Propionamide Frameworks as Potent SARS-CoV-2 Mpro Inhibitor for Treating Coronavirus Disease.” Bioorganic Chemistry, Elsevier, 2026, p. 110102.


BibTeX   Click to copy

@article{alwethaynani2026a,
  title = {Structure-guided optimization of N-(5-((2-oxopropyl) thio)-1, 3, 4-thiadiazol-2-yl) propionamide frameworks as potent SARS-CoV-2 Mpro inhibitor for treating coronavirus disease},
  year = {2026},
  journal = {Bioorganic Chemistry},
  pages = {110102},
  publisher = {Elsevier},
  author = {Alwethaynani, Maher S and Hassan, Reem Nabil and Hussain, Rafaqat and Sarfraz, Hina and Sardar, Asma and Asif, Faisal and Khan, Yousaf and Binsaleh, Ammena Y and Al-Hoshani, Nawal and Mojally, Mariam Ameen and others}
}